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17 天
体外ADME研究——药物Ⅱ相代谢稳定性试验
药物代谢(Drug Metabolism)研究是创新药物研发的重要内容,它不仅决定了创新药物制剂研发的成败,而且与创新药物研发的速度和质量有密切关系。由于肝脏是药物代谢的主要场所,体外代谢模型多以肝脏为基础。目前,研究体外代谢方法主要有:肝微粒体 ...
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