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J-2156:一种有望缓解疼痛的新型化合物
J-2156是一种非肽类化合物,这意味着它不是由氨基酸组成的多肽链。它的结构与生长抑素受体4(sstr4)结合,能够激活下游信号通路,从而发挥缓解疼痛的作用。生长抑素是一种重要的抑制性激素,广泛分布在中枢神经系统和外周组织中,通过负调节多种激素释放和细胞增殖发挥重要作用。
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