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穿膜肽的研究进展:从基础分类到临床应用与未来展望
阳离子肽通过带正电荷的氨基酸(精氨酸、赖氨酸)与细胞膜带负电的磷脂或糖胺聚糖(如硫酸乙酰肝素)结合,诱导膜扰动或直接形成纳米孔,是电荷主导的跨膜机制。代表序列与最新进展: ★ ★ TAT肽(RKKRRQRRR(最短活性肽)或GRKKRRQRRRPPQ(全长片段 ...
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