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PCI-34051对组蛋白去乙酰化酶8的结合机制及远程调控
采用天然质谱法、氢-氘交换质谱法和分子动力学模拟相结合的综合方法,研究PCI-34051对人HDAC8的抑制机制,并与泛抑制剂SAHA进行比较。 探究 HDAC8 抑制剂结合机制与远程调控,助力靶向药物研发 近日,中山大学药学院(第一作者单位)的研究人员 Yuxiang Luo 等人 ...
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