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胆固醇对 EphA2 受体的调控机制:肿瘤研究新突破
本文揭示胆固醇抑制 EphA2 受体自组装及非配体依赖性激活,为肿瘤治疗提供新靶点。 ### 研究背景 受体酪氨酸激酶 EphA2 在多种生理过程中发挥着关键作用,如胚胎发育、神经元可塑性、伤口愈合以及成体上皮组织的稳态维持等。其激活依赖于与 ephrin 配体的结合 ...
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